N-acyliminium intermediates in solid-phase synthesis.

Publikation: Bidrag til tidsskrift › Review › Forskning › fagfællebedømt

Standard

N-acyliminium intermediates in solid-phase synthesis. / Le Quement, Sebastian T.; Petersen, Rico; Meldal, Morten; Nielsen, Thomas E.

I: Biopolymers, Bind 94, Nr. 2, 2010, s. 242-256.

Publikation: Bidrag til tidsskrift › Review › Forskning › fagfællebedømt

Harvard

Le Quement, ST, Petersen, R, Meldal, M & Nielsen, TE 2010, 'N-acyliminium intermediates in solid-phase synthesis.', Biopolymers, bind 94, nr. 2, s. 242-256. https://doi.org/10.1002/bip.21358

APA

Le Quement, S. T., Petersen, R., Meldal, M., & Nielsen, T. E. (2010). N-acyliminium intermediates in solid-phase synthesis. Biopolymers, 94(2), 242-256. https://doi.org/10.1002/bip.21358

Vancouver

Le Quement ST, Petersen R, Meldal M, Nielsen TE. N-acyliminium intermediates in solid-phase synthesis. Biopolymers. 2010;94(2):242-256. https://doi.org/10.1002/bip.21358

Author

Le Quement, Sebastian T. ; Petersen, Rico ; Meldal, Morten ; Nielsen, Thomas E. / N-acyliminium intermediates in solid-phase synthesis. I: Biopolymers. 2010 ; Bind 94, Nr. 2. s. 242-256.

Bibtex

@article{4bd61d25fc844cad9c397535ce7e589c,
title = "N-acyliminium intermediates in solid-phase synthesis.",
abstract = "N-Acyliminium ions are powerful intermediates in synthetic organic chemistry. Examples of their use are numerous in solution-phase synthesis, but there are unmerited few reports on these highly reactive electrophiles in solid-phase synthesis. The present review covers the literature to date and illustrates the methods used to generate N-acyliminium intermediates on solid support and their further elaboration to a range of pharmacologically interesting peptidomimetics, heterocycles, and other small molecules.",
author = "{Le Quement}, {Sebastian T.} and Rico Petersen and Morten Meldal and Nielsen, {Thomas E.}",
year = "2010",
doi = "10.1002/bip.21358",
language = "English",
volume = "94",
pages = "242--256",
journal = "Biopolymers",
issn = "0006-3525",
publisher = "Wiley",
number = "2",

}

RIS

TY - JOUR

T1 - N-acyliminium intermediates in solid-phase synthesis.

AU - Le Quement, Sebastian T.

AU - Petersen, Rico

AU - Meldal, Morten

AU - Nielsen, Thomas E.

PY - 2010

Y1 - 2010

N2 - N-Acyliminium ions are powerful intermediates in synthetic organic chemistry. Examples of their use are numerous in solution-phase synthesis, but there are unmerited few reports on these highly reactive electrophiles in solid-phase synthesis. The present review covers the literature to date and illustrates the methods used to generate N-acyliminium intermediates on solid support and their further elaboration to a range of pharmacologically interesting peptidomimetics, heterocycles, and other small molecules.

AB - N-Acyliminium ions are powerful intermediates in synthetic organic chemistry. Examples of their use are numerous in solution-phase synthesis, but there are unmerited few reports on these highly reactive electrophiles in solid-phase synthesis. The present review covers the literature to date and illustrates the methods used to generate N-acyliminium intermediates on solid support and their further elaboration to a range of pharmacologically interesting peptidomimetics, heterocycles, and other small molecules.

UR - http://www.scopus.com/inward/record.url?scp=77951914699&partnerID=8YFLogxK

U2 - 10.1002/bip.21358

DO - 10.1002/bip.21358

M3 - Review

C2 - 20225296

AN - SCOPUS:77951914699

VL - 94

SP - 242

EP - 256

JO - Biopolymers

JF - Biopolymers

SN - 0006-3525

IS - 2

ER -

ID: 321824844